URB 597 [546141-08-6]

Katalog-Nummer VD-OEIA-0132-10mg

Size : 10mg

Marke : VDM Biochemicals

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Product Specification

  • Appearance
    :

    White solid.

  • CAS Number
    :

    546141-08-6

  • Cat.number
    :

    VD-OEIA-0132

  • Formula
    :

    C20H22N2O3

  • MW
    :

    338.4

  • Purity
    :

    >=98%.

  • Solubility
    :

    50 mM in DMSO.

  • Storage
    :

    +2°C to +8°C. Protect from light.

  • Synonyms
    :

    N/A

  • Size
    :

    10mg, 50mg

SKU: VD-OEIA-0132 Categories: Enzyme Inhibitors, Other Enzyme Inhibitors and Activators

Description

Potent and selective fatty acid amide hydrolase (FAAH) inhibitor (IC50 values are 3 and 5 nM in human liver and rat brain, respectively). Exhibits no significant inhibitory activity against a variety of receptors, ion channels and enzymes, including human cannabinoid receptors and rat monoacylglycerol lipase. Displays antiallodynic and antihyperalgesic activity in an inflammatory pain model.

1.Hohmann et al (2005); Nature 435 1108.
2.Jayamanne et al (2006); Br.J.Pharmacol. 147 281.